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Wopanga ufa wa Amino Tadalafil CAS No.: 385769-84-6 98% chiyero min.kwa zowonjezera zowonjezera

Kufotokozera Kwachidule:

Amino Tadalafil ndi chigawo chofanana ndi Tadalafil, ndi magulu ena ogwira ntchito m'mapangidwe ake amasinthidwa ndi magulu a amino.


Tsatanetsatane wa Zamalonda

Zolemba Zamalonda

Product Parameters

Dzina la malonda

Amino Tadalafil

Dzina lina

(6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[ 3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A -Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dione;(6R,12aR)-2-Amino-6-(benzo[d][1,3] ]dioxol-5-yl) -2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R ,12aR) -2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3] ,4-b]indole-1,4(6H,7H) -dione

CAS No.

385769-84-6

Molecular formula

C21H18N4O4

Kulemera kwa maselo

390.39

Chiyero

98.0%

Maonekedwe

Ufa woyera mpaka woyera

Kugwiritsa ntchito

Zakudya Zowonjezera Zamasamba

Chiyambi cha malonda

Amino Tadalafil ndi chigawo chofanana ndi Tadalafil, ndi magulu ena ogwira ntchito m'mapangidwe ake amasinthidwa ndi magulu a amino.Ndi PDE5 inhibitor ndipo imakhala ndi zotsatira za pharmacological zofanana ndi Tadalafil.Amagwiritsidwa ntchito makamaka pochiza matenda a Erectile Dysfunction (ED).Poyerekeza ndi Tadalafil, Amino Tadalafil ali ndi kagayidwe kakang'ono kamene kali m'thupi, ndipo motero akhoza kukhala ndi zotsatira zokhalitsa.

Mbali

(1) Kusankhidwa kwakukulu: Amino Tadalafil ali ndi kusankha kwakukulu kwa PDE5, ndi kuyanjana kwakukulu kwa PDE5 kusiyana ndi zina za PDE.Izi zikutanthauza kuti Amino Tadalafil amatha kuletsa bwino ntchito ya puloteni ya PDE5, kulimbikitsa kutuluka kwa magazi m'zigawo zoberekera za amuna ndikuwongolera zizindikiro za erectile dysfunction (ED).

(2) Zotsatira zokhalitsa: Amino Tadalafil imakhala ndi kagayidwe kakang'ono kagayidwe kake m'thupi, zomwe zimapangitsa kuti pakhale mphamvu yowonjezereka ya mankhwala, yomwe imakhalapo mpaka maola a 36.Izi zimapangitsa Amino Tadalafil kukhala mankhwala ochizira ED kwa nthawi yayitali, omwe safunikira kutengedwa pafupipafupi.

(3) Zotsatira zochepa: Amino Tadalafil ali ndi zotsatira zochepa poyerekeza ndi Tadalafil, monga kupweteka kwa mutu, ndi kupweteka kwa m'mimba.Chifukwa cha kusankha kwake kwapamwamba, Amino Tadalafil amatha kupewa kuyanjana ndi ma PDE ena, kuchepetsa zotsatira za zotsatira zake.

(4) Chiyembekezo chogwiritsa ntchito kwambiri: Kuphatikiza pa kuchiza ED, Amino Tadalafil angagwiritsidwenso ntchito pochiza matenda ena monga pulmonary arterial hypertension.Izi zimapangitsa Amino Tadalafil kukhala ndi chiyembekezo chogwiritsa ntchito mtsogolo.

Mapulogalamu

Amino Tadalafil ndi gulu lomwe linapangidwa m'zaka zaposachedwa, lomwe lili ndi dongosolo lofanana ndi Tadalafil, koma magulu ena omwe ali m'magulu ake amasinthidwa ndi magulu a amino.Pakalipano, Amino Tadalafil sanavomerezedwe kuti agwiritsidwe ntchito pachipatala, choncho ntchito yake m'chipatala ndi yochepa.Komabe, kafukufuku wina wasonyeza kuti mankhwalawa ali ndi kuthekera kwakukulu kogwiritsa ntchito.

Amino Tadalafil ndi PDE5 inhibitor, yomwe ili ndi zotsatira zofanana za mankhwala monga Tadalafil.Ikhoza kusintha zizindikiro za erectile dysfunction (ED) mwa kulimbikitsa kutuluka kwa magazi mu ziwalo zoberekera za amuna poletsa ntchito ya PDE5 enzyme.Poyerekeza ndi Tadalafil, Amino Tadalafil ali ndi kagayidwe kake kake kagayidwe m'thupi, zomwe zingakhale ndi zotsatira zokhalitsa.Izi zimapangitsa Amino Tadalafil kukhala ndi kuthekera kwakukulu pakuchiza ED.

Kuphatikiza apo, Amino Tadalafil itha kugwiritsidwanso ntchito pochiza matenda ena, monga pulmonary arterial hypertension.Kafukufuku wina wasonyeza kuti PDE5 inhibitors amatha kufutukula mitsempha ya m'mapapo, potero kusintha zizindikiro za odwala ndi pulmonary arterial hypertension.Chifukwa Amino Tadalafil ali ndi mphamvu yofananira yamankhwala monga Tadalafil, itha kugwiritsidwanso ntchito pochiza matenda oopsa a pulmonary arterial hypertension.

Ponseponse, Amino Tadalafil ali ndi kuthekera kwakukulu kogwiritsa ntchito, koma mayeso ochulukirapo azachipatala amafunikira kuti adziwe chitetezo chake ndi mphamvu zake.Ngati mayeserowa apereka zotsatira zabwino, Amino Tadalafil akhoza kukhala mankhwala atsopano ochizira ED ndi pulmonary arterial hypertension, kupereka njira zambiri zothandizira madokotala ndi odwala.


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