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malonda

Wopanga ufa wa Amino Tadalafil Nambala ya CAS: 385769-84-6 98% kuyera pang'ono kwa zosakaniza zowonjezera

Kufotokozera Kwachidule:

Amino Tadalafil ndi chinthu chofanana ndi Tadalafil, ndipo magulu ena ogwira ntchito m'mapangidwe ake amalowedwa m'malo ndi magulu a amino.


Tsatanetsatane wa Zamalonda

Ma tag a Zamalonda

Kanema wa Zamalonda

Magawo a Zamalonda

Dzina la chinthu

Amino Tadalafil

Dzina lina

(6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A-Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dion e;(6R,12aR)-2-Amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R,12aR)-2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4(6H,7H)-dione

Nambala ya CAS

385769-84-6

Fomula ya maselo

C21H18N4O4

Kulemera kwa maselo

390.39

Chiyero

98.0%

Maonekedwe

Ufa woyera mpaka woyera pang'ono

Kugwiritsa ntchito

Zakudya Zowonjezera Zakudya

Chiyambi cha malonda

Amino Tadalafil ndi mankhwala atsopano, ochokera ku tadalafil, omwe akutchuka kwambiri pankhani ya erectile dysfunction (ED). Amaphatikiza amino acid ndi tadalafil, choletsa cha PDE5 chovomerezeka ndi FDA chomwe chimagwiritsidwa ntchito makamaka pochiza ED. Imagwira ntchito powonjezera kuyenda kwa magazi kupita ku mbolo, zomwe zimathandiza amuna kukwaniritsa ndikusunga mbewa. Koma ma amino acid, amatenga gawo lofunikira kwambiri pa ntchito zosiyanasiyana za thupi, kuphatikizapo kupanga mapuloteni, omwe ndi zomangira minofu ndi ziwalo. Kuphatikiza kwa zosakaniza ziwirizi kwapangidwa kuti kuwonjezere mphamvu ya Tadalafil pochiza ED. Ndipo amino Tadalafil ndi mtundu wabwino kwambiri wokhala ndi mphamvu zodabwitsa, zomwe zimapangitsa kuti ntchito yake ikhale yosiyana komanso yosinthasintha. Kapangidwe kake ka mankhwala kamakhala kofanana ndi Tadalafil, koma kudzera mu kuyambitsa magulu a amino, imapeza makhalidwe apadera omwe amaipangitsa kukhala yodziwika bwino m'dziko la mankhwala. Monga tadalafil, Amino Tadalafil imagwira ntchito poletsa phosphodiesterase 5 (PDE5), enzyme yomwe imayang'anira kuphwanya guanosine monophosphate (cGMP) m'thupi. cGMP ndi mankhwala achilengedwe omwe amalimbikitsa kumasuka kwa mitsempha yamagazi, motero amawonjezera kuyenda kwa magazi. Mwa kuletsa PDE5, amino Tadalafil imatsimikizira kuti cGMP ikuwonjezeka, motero imakulitsa kufalikira kwa magazi ndikukweza kuyenda kwa magazi. Kuphatikiza apo, ofufuza afufuza momwe ingathandizire kuchiza benign prostatic hyperplasia (BPH) mwa kulimbikitsa kuyenda kwa magazi kupita ku prostate.

Mbali

(1) Kuyera Kwambiri: Amino Tadalafil imatha kupeza zinthu zoyera kwambiri kudzera mu njira zopangira zinthu zoyeretsera. Kuyera Kwambiri kumatanthauza kupezeka bwino kwa bioavailability komanso kuchepetsa zotsatirapo zoyipa.

(2) Chitetezo: Chitetezo chapamwamba, zotsatirapo zochepa zoyipa.

(3) Kukhazikika: Amino Tadalafil ili ndi kukhazikika kwabwino ndipo imatha kusunga ntchito yake ndi mphamvu zake pansi pa malo osiyanasiyana komanso malo osungiramo zinthu zosiyanasiyana.

Mapulogalamu

Amino Tadalafil ndi mankhwala oletsa PDE5 omwe ali ndi zotsatira zofanana ndi tadalafil. Mwa kuphatikiza ma amino acid ndi tadalafil, amino Tadalafil imaganiziridwa kuti ndi yothandiza kwambiri pochiza vuto la erectile kusiyana ndi tadalafil yokha. Ma amino acid angathandize kupititsa patsogolo kuyenda kwa magazi ndikuthandizira kugwira ntchito bwino kwa mankhwala. Kuphatikiza apo, imatha kukonza zizindikiro za erectile dysfunction (ED) poletsa ntchito ya enzyme ya PDE5 kuti magazi aziyenda bwino m'ziwalo zoberekera za amuna. Poyerekeza ndi tadalafil, amino Tadalafil imaphikidwa pang'onopang'ono m'thupi ndipo imatha kukhala ndi zotsatira zokhalitsa. Izi zimapatsa amino Tadalafil mwayi waukulu pochiza ED.


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