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Wopanga ufa wa Coluracetam CAS No.: 135463-81-9 99% chiyero min.kwa zowonjezera zowonjezera

Kufotokozera Kwachidule:

Coluracetam ndi membala wa banja la racetam la mankhwala a nootropic ndipo amadziwikanso kuti MKC-231.Idapangidwa ndi Kobe Pharmaceutical Company ku Japan ndi cholinga chochiza AD ndi kusokonezeka kwa chidziwitso.


Tsatanetsatane wa Zamalonda

Zolemba Zamalonda

Product Parameters

Dzina la malonda

Coluracetam

Dzina lina

MKC-231;

2-oxo-N-(5,6,7,8-tetrahydro-2,3-dimethyl-furo[2,3-b]quinolin-4-yl) -1-pyrrolidineacetamide

CAS No.

135463-81-9

Molecular formula

Chithunzi cha C19H23N3O3

Kulemera kwa maselo

341.4

Chiyero

99.0%

Maonekedwe

White ufa

Kugwiritsa ntchito

Zakudya Zowonjezera Zamasamba

Chiyambi cha malonda

Coluracetam ndi membala wa banja la racetam la mankhwala a nootropic ndipo amadziwikanso kuti MKC-231.Idapangidwa ndi Kobe Pharmaceutical Company ku Japan ndi cholinga chochiza AD ndi kusokonezeka kwa chidziwitso.

Njira yeniyeni ya Coluracetam sichimveka bwino, koma imakhulupirira kuti imagwira ntchito makamaka pokonza dongosolo la cholinergic.Zimaganiziridwa kuti zimawonjezera kuchuluka kwa acetylcholine, neurotransmitter yofunika kwambiri muubongo yomwe imagwirizana kwambiri ndi kuphunzira ndi kukumbukira ntchito.Coluracetam ikhoza kukwaniritsa izi mwa kuonjezera chiwerengero ndi ntchito za onyamula choline, zomwe zimapangitsa kuti acetylcholine atulutsidwe komanso kupititsa patsogolo kufalikira kwa zizindikiro pakati pa neuroni.

Ngakhale kuti kafukufuku wa Coluracetam akadali wochepa, mayesero ena oyambirira ndi maphunziro a zinyama awonetsa kuti zotsatira za neuroprotective ndi chidziwitso-zingakhale zowonjezera.Kafukufuku wina wapeza kuti Coluracetam ili ndi kusintha kwina kwa kukumbukira kukumbukira mu zitsanzo za AD.

Pankhani ya kafukufuku wachipatala, maphunziro a Coluracetam makamaka amayang'ana pa kuyesa kwa nyama ndi mayesero oyambirira a anthu.Kafukufuku wambiri ndi umboni ndizofunikira kuti mudziwe chitetezo chake ndi mphamvu zake mwa anthu.Pakalipano, Coluracetam sinavomerezedwe kuti igwiritsidwe ntchito kuchipatala, koma imagwiritsidwa ntchito kwambiri ngati mankhwala a nootropic pofuna kupititsa patsogolo chidziwitso m'mayiko ena.

Ponena za chitetezo, pali kafukufuku wochepa wopezeka pa zotsatirapo ndi zoopsa za nthawi yaitali za Coluracetam.Malingana ndi chidziwitso chamakono, Coluracetam nthawi zambiri amaonedwa kuti ndi yotetezeka, komabe amalangizidwa kuti akambirane ndi katswiri wa zaumoyo, makamaka ngati muli ndi thanzi labwino kapena mukumwa mankhwala ena, musanagwiritse ntchito.

Mwachidule, Coluracetam ndi mankhwala a nootropic omwe akuphunziridwa chifukwa cha kuthekera kwake pochiza AD ndi kuwonongeka kwa chidziwitso.Ngakhale kafukufuku wina woyambirira akuwonetsa kupititsa patsogolo kwachidziwitso ndi zotsatira za neuroprotective, maphunziro ochulukirapo akufunika kuti atsimikizire momwe zimagwirira ntchito komanso chitetezo chake.

Mbali

(1) Kuyera Kwambiri: Coluracetam imakonzedwa pogwiritsa ntchito njira zotsogola ndi kupanga, kuonetsetsa kuti pakhale chiyero chapamwamba.Kuyera kotereku kumathandizira kuti bioavailability ikhale yabwino komanso kumachepetsa kuchitika kwa zoyipa.

(2) Chitetezo: Coluracetam imatengedwa kuti ndi yotetezeka kuti anthu adye.Kafukufuku wambiri wasonyeza kuti ali ndi kawopsedwe kakang'ono komanso zotsatira zake zochepa pamlingo wovomerezeka.

(3) Kukhazikika: Kukonzekera kwa Coluracetam kumasonyeza kukhazikika kwabwino, kusunga ntchito zawo ndi zogwira mtima pansi pa zochitika zosiyanasiyana zachilengedwe ndi zosungirako.Kukhazikika kumeneku kumatsimikizira kugwira ntchito kosasinthasintha komanso kodalirika pakapita nthawi.

(4) Kuthamanga Mofulumira: Coluracetam imatengedwa mosavuta ndi thupi la munthu.Akamadya, amalowa m'magazi mwamsanga kudzera m'matumbo a m'mimba ndikugawira bwino ku ziwalo zosiyanasiyana ndi ziwalo, zomwe zimathandizira zotsatira zake.

(5) Kupititsa patsogolo Chidziwitso: Coluracetam imadziwika kuti imatha kupititsa patsogolo chidziwitso, kuphatikizapo kusintha kwa kukumbukira, kuphunzira, ndi kuganizira.Nthawi zambiri amafunidwa ndi anthu omwe akufuna kukulitsa luso lawo lamalingaliro.

(6) Zotsatira za Neuroprotective: Kafukufuku akuwonetsa kuti Coluracetam ikhoza kukhala ndi mphamvu zoteteza ubongo, zomwe zingathandize kuteteza kuchepa kwa chidziwitso chokhudzana ndi ukalamba ndikuthandizira thanzi laubongo lonse.

(7) Chithandizo Chothekera cha Kusokonezeka Maganizo: Coluracetam imasonyeza lonjezo ngati njira yochizira matenda a chidziwitso, monga matenda a Alzheimer's and other neurodegenerative.Komabe, kufufuza kwina kumafunika kuti timvetsetse bwino momwe zimagwirira ntchito pochiza mikhalidwe imeneyi.

Mapulogalamu

Coluracetam ikugwiritsidwa ntchito pazochitika zosiyanasiyana ndipo ikuwonetsa chiyembekezo chamtsogolo.Amagwiritsidwa ntchito makamaka ngati chowonjezera chazidziwitso, chomwe chimafunidwa ndi anthu omwe akufuna kukonza kukumbukira kwawo, kuyang'ana, ndi luso la kuphunzira.Kuthekera kwa gululi kuwongolera dongosolo la cholinergic kumakhulupirira kuti kumathandizira kukulitsa chidziwitso.

Kuphatikiza pa ntchito zake zamakono, Coluracetam yawonetsa kuthekera kochiza matenda a neurodegenerative monga matenda a Alzheimer's ndi kuwonongeka kwa chidziwitso.Kafukufuku akuwonetsa kuti Coluracetam ikhoza kukhala ndi mphamvu zoteteza ubongo, zomwe zimapangitsa kuti ikhale yochititsa chidwi kuti ifufuze mopitilira muzochitika izi.Komabe, maphunziro owonjezera ndi mayesero azachipatala amafunikira kuti adziwe momwe angagwiritsire ntchito bwino, chitetezo chake, komanso njira zoyenera zogwiritsira ntchito m'machipatala.

Chiwerengero cha anthu okalamba chawonjezera kufunika kochitapo kanthu komwe kungachepetse kuchepa kwa chidziwitso chokhudzana ndi ukalamba.Zotsatira za neuroprotective za Coluracetam komanso kuthekera kothandizira njira zokonzetsera ma neural zimapangitsa kukhala njira yosangalatsa yofufuzira pothana ndi kuchepa kwa chidziwitso komwe kumakhudzana ndi ukalamba.

Kuphatikiza apo, kafukufuku woyambirira akuwonetsa kuti Coluracetam ikhoza kukhala ndi phindu pazovuta zamalingaliro monga kukhumudwa ndi nkhawa.Komabe, maphunziro owonjezereka amafunikira kuti awone momwe angagwiritsire ntchito bwino ndikukhazikitsa njira zochiritsira zoyenera pazizindikirozi.

Kuthekera kwa Coluracetam kumafikiranso ku mapulogalamu a neurorehabilitation.Kuthekera kwake kukulitsa ma signature a neuronal komanso kuthandizira njira zokonzetsera ma neural kumapangitsa kuti ikhale yoyenera kugwiritsidwa ntchito pokonzanso anthu omwe akuvulala muubongo kapena zikwapu.

Ngakhale kuti Coluracetam imasonyeza lonjezano muzogwiritsira ntchito zosiyanasiyana, ndikofunika kutsindika kufunikira kwa kufufuza kwina, kutsimikizira mphamvu zake, chitetezo, ndi ndondomeko zogwiritsira ntchito bwino.Zivomerezo zovomerezeka ziyeneranso kufunikira kuti zigwiritsidwe ntchito pachipatala pazisonyezero zinazake.


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