Wopanga ufa wa Coluracetam Nambala ya CAS: 135463-81-9 99% chiyero cha zosakaniza zowonjezera
Kanema wa Zamalonda
Magawo a Zamalonda
| Dzina la chinthu | Coluracetam |
| Dzina lina | MKC-231; 2-oxo-N-(5,6,7,8-tetrahydro-2,3-dimethyl-furo[2,3-b]quinolin-4-yl)-1-pyrrolidineacetamide |
| Nambala ya CAS | 135463-81-9 |
| Fomula ya maselo | C19H23N3O3 |
| Kulemera kwa maselo | 341.4 |
| Chiyero | 99.0% |
| Maonekedwe | Ufa woyera |
| Kugwiritsa ntchito | Zakudya Zowonjezera Zakudya |
Chiyambi cha malonda
Coluracetam, yomwe ndi membala wa banja la racemate la mankhwala a nootropic, omwe amadziwikanso kuti MKC-231, ndi mankhwala a nootropic omwe ali ndi zotsatira zowonjezera chidziwitso komanso zoteteza mitsempha. Coluracetam imagwira ntchito posintha dongosolo la cholinergic. Akuganiza kuti imawonjezera kuchuluka kwa acetylcholine, neurotransmitter yofunika kwambiri muubongo yolumikizidwa kwambiri ndi kuphunzira ndi ntchito zokumbukira. Coluracetam imachita izi powonjezera kuchuluka ndi ntchito za zonyamula choline, motero imakulitsa kutulutsidwa kwa acetylcholine ndikuwongolera kulumikizana pakati pa ma neuron. Kafukufuku wina woyambirira komanso wa nyama akuwonetsa kuti Coluracetam ili ndi mphamvu zoteteza mitsempha komanso zolimbikitsa chidziwitso. Kafukufuku wina wapeza kuti Coluracetam ili ndi zotsatira zina zabwino pa kuwonongeka kwa kukumbukira m'mamodeli a AD.
Mbali
(1) Kuyera kwambiri: Coluracetam imakonzedwa pogwiritsa ntchito njira zapamwamba zochotsera ndi kupanga kuti zitsimikizire kuti ndi yoyera kwambiri. Kuyera kwakukulu kumeneku kumathandiza kukonza kupezeka kwa bioavailability ndikuchepetsa kuchitika kwa zotsatira zoyipa.
(2) Chitetezo: Coluracetam imaonedwa kuti ndi yotetezeka kwa anthu. Kafukufuku wambiri wasonyeza kuti ili ndi poizoni wochepa komanso zotsatirapo zochepa mkati mwa mlingo woyenera.
(3) Kukhazikika: Mankhwala a Coluracetam amakhala okhazikika bwino ndipo amatha kusunga ntchito yawo komanso kugwira ntchito bwino m'malo osiyanasiyana komanso m'malo osungiramo zinthu zosiyanasiyana. Kukhazikika kumeneku kumatsimikizira kuti ntchito yake ndi yokhazikika komanso yodalirika kwa nthawi yayitali.
Mapulogalamu
Coluracetam pakadali pano imagwiritsidwa ntchito m'njira zosiyanasiyana ndipo ikuwonetsa chiyembekezo chabwino chamtsogolo. Imagwiritsidwa ntchito makamaka ngati chowonjezera chowonjezera pazakudya ndipo imafunidwa ndi anthu omwe akufuna kukonza kukumbukira, kuyang'ana kwambiri, komanso luso lophunzira. Kuthekera kwa mankhwalawa kusintha dongosolo la cholinergic kumaganiziridwa kuti kumathandizira pakukula kwa chidziwitso. Kuphatikiza apo, kafukufuku akuwonetsa kuti Coluracetam ikhoza kukhala ndi mphamvu zoteteza mitsempha zomwe zingathandize kupewa kuchepa kwa chidziwitso chokhudzana ndi ukalamba ndikuthandizira thanzi lonse la ubongo.












