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Wopanga ufa wa Compound 7P Nambala ya CAS: 1890208-58-8 99% kuyera kwa mphindi zochepa kwa zosakaniza zowonjezera

Kufotokozera Kwachidule:

Compound 7p yawonetsedwa kuti imayambitsa kukula kwa ma axon a GAP-43-positive mu chitsanzo cha nyama cha kuvulala kwa mitsempha ya optic, zomwe zikusonyeza kuti ntchito yokulira ya neurite ya compound 7p mu vitro imasintha kukhala kukulitsa kwa axon regeneration mu vivo.


Tsatanetsatane wa Zamalonda

Ma tag a Zamalonda

Kanema wa Zamalonda

Magawo a Zamalonda

Dzina la chinthu

Pawiri 7P

Dzina lina

Compound7P;2-[(2-methoxyphenyl)[(4-methylphenyl)sulfonyl]amino]-N-(4-methoxy-3-pyridinyl)acetamide;

2-(N-(2-methoxyphenyl)-4-methylphenylsulfonamido)-N-(4-methoxypyridin-3-yl)acetamide

Nambala ya CAS

1890208-58-8

Fomula ya maselo

C22H23N3O5S

Kulemera kwa maselo

441.51

Chiyero

99.0%

Maonekedwe

Ufa woyera

Kugwiritsa ntchito

Mankhwala oletsa kutupa (Nootropic)

Chiyambi cha malonda

Compound 7P imatanthauza chinthu chachilengedwe chomwe chili ndi maatomu asanu ndi awiri a kaboni. Mu organic chemistry, kaboni ndi chinthu chofunikira kwambiri chifukwa chimatha kupanga maubwenzi okhazikika ndi maatomu ena, kuphatikiza maatomu a kaboni, kuti apange mamolekyu ovuta. Mamolekyu amenewa amatha kukhala ndi zinthu zosiyanasiyana komanso ntchito zosiyanasiyana, zomwe zimapangitsa kuti ma carbon-based compounds akhale zinthu zomangira moyo. Mu zitsanzo za nyama zomwe zimavulala ndi mitsempha ya optic, compound 7p idawonetsedwa kuti imayambitsa kukula kwa ma axon a GAP-43-positive, zomwe zikusonyeza kuti ntchito ya kukula kwa neurite ya compound 7p in vitro imasintha kukhala kukulitsa kwa axonal regeneration in vivo. Compound 7P powder ndi ufa woyera mpaka woyera womwe umapangidwa ngati tandem compound kuti uzindikire ma dual-acting thromboxane receptor antagonist inhibitors. Ndipotu, compound 7p idawonetsa kusankha kwa prostaglandin I2 synthase (PTGIS, CYP8A1) poyerekeza ndi thromboxane synthase (CYP5A1). Nootropic compound 7P powder imalimbikitsa kukula kwa ma axon a Gap-43-positive, motero imalimbikitsa axonal regeneration m'thupi. Complex 7p yapamwamba kwambiri yapangidwa kuti ipangitse kuti zinthu zizigwirizana bwino, kusintha momwe munthu akumvera komanso kulimbana ndi kutopa. Imaletsanso kukhuthala kwa ubongo komanso imathandiza kulimbana ndi kuwonongeka kwa ubongo komwe kumachitika chifukwa chomwa mowa.

Mbali

结构图

(1) Kuyera Kwambiri: Compound 7P imatha kupeza zinthu zoyera kwambiri kudzera mu njira zopangira zoyengedwa bwino. Kuyera Kwambiri kumatanthauza kupezeka bwino kwa bioavailability komanso kuchepetsa zotsatira zoyipa.

(2) Chitetezo: Compound 7P yatsimikiziridwa kuti ndi yotetezeka ku thupi la munthu.

(3) Kukhazikika: Compound 7P ili ndi kukhazikika kwabwino ndipo imatha kusunga ntchito yake ndi mphamvu zake pansi pa malo osiyanasiyana komanso malo osungiramo zinthu zosiyanasiyana.

Mapulogalamu

Compound 7p imathandizira kukula kwa ma neuron oyambira omwe amakula ochokera ku hippocampus, cerebral cortex, ndi retina ndipo imayambitsa kukonzanso kwa mitsempha ya optic mu zitsanzo za nyama zomwe zimavulala ndi mitsempha ya optic. Imathandizanso kulumikizana bwino, imachiritsa kuwonongeka kwa ubongo komwe kumachitika chifukwa cha mowa, komanso imaletsa okosijeni kuzungulira ubongo. Imathandizanso kukonza malingaliro ndikulimbana ndi kutopa.


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