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RU58841 wopanga ufa CAS No.: 154992-24-2 99.0% chiyero min.kwa zowonjezera zowonjezera

Kufotokozera Kwachidule:

RU58841 (yomwe imadziwikanso kuti RU-58841) ndi mankhwala, RU58841 amapikisana ndi dihydrotestosterone kuti asunge miyeso ya DHT mkati mwanthawi zonse, potero imayendetsa kakulidwe ka tsitsi.Zimapangitsa kutembenuka kwa tsitsi latsopano kukhala ma follicle a tsitsi la anagen polowa mu gawo la anagen.


Tsatanetsatane wa Zamalonda

Zolemba Zamalonda

Product Parameters

Dzina la malonda

4--[3-(4-Hydroxybutyl)-4,4-dimethyl-2,5-dioxo-1-imidazolidinyl]-2-(trifluoromethyl)benzonitrile

Dzina lina

RU58841

CAS No.

154992-24-2

Molecular formula

Chithunzi cha C17H18F3N3O3

Kulemera kwa maselo

369.34

Chiyero

99.0%

Maonekedwe

ufa woyera

Kulongedza

1kg/chikwama

Kugwiritsa ntchito

Kulitsani tsitsi

Chiyambi cha malonda

RU58841 (yomwe imadziwikanso kuti RU-58841) ndi mankhwala, RU58841 amapikisana ndi dihydrotestosterone kuti asunge miyeso ya DHT mkati mwanthawi zonse, potero imayendetsa kakulidwe ka tsitsi.Zimapangitsa kutembenuka kwa tsitsi latsopano kukhala ma follicle a tsitsi la anagen polowa mu gawo la anagen.Kulola ma follicles owonongeka nthawi kuti abwerere ku gawo lakukula bwino kumathandiza maselo kuti achire.Zimawonjezeranso kutuluka kwa magazi ku follicles zowonongeka ndikuwathandiza kuti abwererenso.Kumbali inayi, RU58841 (RU-58841) imagwira ntchito pomanga ma androgen receptors muzitsulo za tsitsi.Chifukwa chake ma androgens alibe mwayi womanga ndikuyamba kuchitapo kanthu kwa androgenetic alopecia ndikuyamba njira yotchedwa miniaturization.Zawonetsedwa kuti zimasokoneza uthenga wotayika tsitsiwu m'deralo kuti kukula kwa tsitsi kupitirire.

Mbali

(1) Ingalepheretse kutayika kwa tsitsi: RU58841 ndi inhibitor yapadera ya hormone, yomwe ingalepheretse kuphatikiza kwa androgen ndi scalp follicle cell cell, potero kuchepetsa chiopsezo cha tsitsi.
(2) Mayamwidwe abwino: RU58841 ili ndi kachidutswa kakang'ono ka maselo, kapangidwe kosavuta, ndipo ndi kosavuta kuyamwa.Imatha kulowa mwachangu m'thupi ndikugwira ntchito munthawi yochepa.
(3) Kusankhidwa kwakukulu kwa androgen: RU58841 ikhoza kuletsa mwachisawawa zochita za androgen popanda kukhudza mahomoni ena.
(4) Nthawi yayitali yochitapo kanthu: RU58841 imakhala ndi theka la moyo wautali m'thupi, imatha kuletsa mosalekeza zotsatira za androgen, ndipo nthawi yogwira ntchito imatha kukhala maola 48.
(5) Kuyera Kwambiri: Kupyolera mu m'zigawo zachilengedwe ndi kupanga bwino, chitukuko cha RU58841 chikhoza kupeza zinthu zoyera kwambiri.

Mapulogalamu

Mu kafukufuku ndi mayesero a zachipatala, RU58841 yasonyezedwa kuti iwonjezere kuchuluka kwa maselo obwerezabwereza m'maselo a stromal, kuonjezera kuchuluka kwa maselo m'maselo akunja a mizu ndikuwonjezera tsitsi la tsitsi ndi kachulukidwe ka tsitsi, kotero RU58841 ndi mankhwala ofufuza pofuna kuchiza androgenetic alopecia.Mfundo yaikulu yogwirira ntchito ndikuletsa kuphatikiza kwa DHT ndi AR ya follicles ya tsitsi, yomwe nthawi zambiri imagwiritsidwa ntchito pochiza kutayika kwa tsitsi ndi kutayika tsitsi.


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