Wopanga ufa wa RU58841 Nambala ya CAS: 154992-24-2 99.0% kuyera pang'ono kwa zosakaniza zowonjezera
Magawo a Zamalonda
| Dzina la chinthu | 4-[3-(4-Hydroxybutyl)-4,4-dimethyl-2,5-dioxo-1-imidazolidinyl]-2-(trifluoromethyl)benzonitrile |
| Dzina lina | RU58841 |
| Nambala ya CAS | 154992-24-2 |
| Fomula ya maselo | C17H18F3N3O3 |
| Kulemera kwa maselo | 369.34 |
| Chiyero | 99.0% |
| Maonekedwe | ufa woyera |
| Kulongedza | 1kg/thumba |
| Kugwiritsa ntchito | Kukulitsa tsitsi |
Chiyambi cha malonda
RU58841 (yomwe imadziwikanso kuti RU-58841) ndi mankhwala opangidwa ndi RU58841, omwe amapikisana ndi dihydrotestosterone kuti asunge milingo ya DHT mkati mwa nthawi zonse, motero amayang'anira kukula kwa tsitsi. Zimathandizira kusintha kwa ma follicle atsopano a tsitsi kukhala ma follicle a tsitsi la anagen polowa mu gawo la anagen. Kulola ma follicle owonongeka nthawi yobwerera ku gawo labwinobwino la kukula kumathandiza maselo kuchira. Zimawonjezeranso kuyenda kwa magazi kupita ku ma follicle owonongeka ndikuwathandiza kubwereranso. Kumbali inayi, RU58841 (RU-58841) imagwira ntchito pomangirira ku ma androgen receptors mu ma follicle a tsitsi. Chifukwa chake ma androgen alibe mwayi womangirira ndikuyamba njira ya androgenetic alopecia ndikuyamba njira yotchedwa miniaturization. Zawonetsedwa kuti zimasokoneza uthenga wotayika tsitsi kuti kukula kwabwinobwino kwa tsitsi kupitirire.
Mbali
(1) Imatha kuletsa kutayika kwa tsitsi: RU58841 ndi mankhwala apadera oletsa mahomoni, omwe amatha kuletsa kuphatikiza kwa maselo a androgen ndi follicle ya tsitsi la scalp, potero amachepetsa chiopsezo cha kutayika kwa tsitsi.
(2) Kuyamwa bwino: RU58841 ili ndi kulemera kochepa kwa mamolekyulu, kapangidwe kosavuta, ndipo ndi kosavuta kuyamwa. Imatha kulowa m'thupi mwachangu ndikugwira ntchito mwachangu.
(3) Kusankha kwambiri androgen: RU58841 ikhoza kuletsa ntchito ya androgen popanda kukhudza mahomoni ena.
(4) Nthawi yayitali yogwira ntchito: RU58841 imakhala ndi theka la moyo m'thupi, imatha kuletsa mphamvu ya androgen nthawi zonse, ndipo nthawi yogwira ntchito imatha kukhala maola 48.
(5) Kuyera Kwambiri: Kudzera mu kuchotsa zinthu zachilengedwe ndi njira zopangira zinthu zabwino, kupanga RU58841 kumatha kupeza zinthu zoyera kwambiri.
Mapulogalamu
Mu kafukufuku ndi mayeso azachipatala, RU58841 yawonetsedwa kuti imawonjezera kuchuluka kwa maselo m'maselo a stromal, imawonjezera kuchulukana kwa maselo m'maselo akunja kwa mizu ndikuwonjezera kukula kwa tsitsi ndi kuchuluka kwa tsitsi, kotero RU58841 ndi mankhwala ofufuza ochizira androgenetic alopecia. Mfundo yayikulu yogwira ntchito ndikuletsa kuphatikiza kwa DHT ndi AR kwa ma follicles a tsitsi, omwe nthawi zambiri amagwiritsidwa ntchito pochiza mavuto otaya tsitsi ndi kutaya tsitsi.












